Molecules, Vol. 24, Pages 2420: Suitability Evaluation of LaNi5 as Hydrogen-Storage-Alloy Actuator by In-Situ Displacement Measurement during Hydrogen Pressure Change Molecules doi: 10.3390/molecules24132420 Authors: Kenta Goto Tomoyuki Hirata Isao Yamamoto Wataru Nakao The swelling ability of LaNi5 for application to hydrogen-storage-alloy (HSA) actuator is discussed through the measurement of the swelling ratio in hydrogen. The HSA actuator is driven by hydrogen pressure change...
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Molecules, Vol. 24, Pages 2419: Hydrated Zinc Borates and Their Industrial Use Molecules doi: 10.3390/molecules24132419 Authors: Schubert Zinc borates are important chemical products having industrial applications as functional additives in polymers, bio-composites, paints and ceramics. Of the thirteen well documented hydrated binary zinc borates, Zn[B3O4(OH)3] (2ZnO∙3B2O3∙3H2O) is manufactured in the largest quantity and is known as an article of commerce as 2ZnO∙3B2O3∙3.5H2O. Other...
Sun Jun 30, 2019 03:00
Molecules, Vol. 24, Pages 2418: Synthesis, Molecular Docking Analysis, and Carbonic Anhydrase Inhibitory Evaluations of Benzenesulfonamide Derivatives Containing Thiazolidinone Molecules doi: 10.3390/molecules24132418 Authors: Zhang Yin Li Wang Wu Wang Liu Cheng To find novel human carbonic anhydrase (hCA) inhibitors, we synthesized thirteen compounds by combining thiazolidinone with benzenesulfonamide. The result of the X-ray single-crystal diffraction experiment...
Sun Jun 30, 2019 03:00
Molecules, Vol. 24, Pages 2415: Breakthroughs in Medicinal Chemistry: New Targets and Mechanisms, New Drugs, New Hopes–5 Molecules doi: 10.3390/molecules24132415 Authors: Arduino A. Mangoni Jean Jacques Vanden Eynde Josef Jampilek Dimitra Hadjipavlou-Litina Hong Liu Jóhannes Reynisson Maria Emília Sousa Paula A. C. Gomes Katalin Prokai-Tatrai Tiziano Tuccinardi Jean-Marc Sabatier F. Javier Luque Jarkko Rautio Rafik Karaman M. Helena Vasconcelos Sandra...
Sun Jun 30, 2019 03:00
Molecules, Vol. 24, Pages 2416: G-Quadruplex-Based Fluorescent Turn-On Ligands and Aptamers: From Development to Applications Molecules doi: 10.3390/molecules24132416 Authors: Mubarak I. Umar Danyang Ji Chun-Yin Chan Chun Kit Kwok Guanine (G)-quadruplexes (G4s) are unique nucleic acid structures that are formed by stacked G-tetrads in G-rich DNA or RNA sequences. G4s have been reported to play significant roles in various cellular events in both macro- and micro-organisms. The...
Sun Jun 30, 2019 03:00
Molecules, Vol. 24, Pages 2417: LIR Motif-Containing Hyperdisulfide β-Ginkgotide is Cytoprotective, Adaptogenic, and Scaffold-Ready Molecules doi: 10.3390/molecules24132417 Authors: Dutta Huang To Tam Grafting a bioactive peptide onto a disulfide-rich scaffold is a promising approach to improve its structure and metabolic stability. The ginkgo plant-derived β-ginkgotide β-gB1 is a highly unusual molecule: Small, hyperdisulfide, and found only in selected...
Sun Jun 30, 2019 03:00
Molecules, Vol. 24, Pages 2414: A Ligand-Based Virtual Screening Method Using Direct Quantification of Generalization Ability Molecules doi: 10.3390/molecules24132414 Authors: Weixing Dai Dianjing Guo Machine learning plays an important role in ligand-based virtual screening. However, conventional machine learning approaches tend to be inefficient when dealing with such problems where the data are imbalanced and features describing the chemical characteristic of ligands are high-dimensional....
Sun Jun 30, 2019 03:00
Molecules, Vol. 24, Pages 2412: Euphosantianane E–G: Three New Premyrsinane Type Diterpenoids from Euphorbia sanctae-catharinae with Contribution to Chemotaxonomy Molecules doi: 10.3390/molecules24132412 Authors: Abdelsamed I. Elshamy Tarik A. Mohamed Saud L. Al-Rowaily Ahmed M. Abd-ElGawad Basharat A. Dar Abdelaaty A. Shahat Mohamed-Elamir F. Hegazy Euphorbia species were widely used in traditional medicines for the treatment of several diseases. From the aerial parts...
Sat Jun 29, 2019 03:00
Molecules, Vol. 24, Pages 2413: A Comparative Study of the Anticancer Activity and PARP-1 Inhibiting Effect of Benzofuran–Pyrazole Scaffold and Its Nano-Sized Particles in Human Breast Cancer Cells Molecules doi: 10.3390/molecules24132413 Authors: Manal M. Anwar Somaia S. Abd El-Karim Ahlam H. Mahmoud Abd El-Galil E. Amr Mohamed A. Al-Omar Breast cancer is considered the most common and deadly cancer among women worldwide. Nanomedicine has become extremely attractive in the...
Sat Jun 29, 2019 03:00
Molecules, Vol. 24, Pages 2410: Intracellular Accumulation as an Indicator of Cytotoxicity to Screen Hepatotoxic Components of Chelidonium majus L. by LC–MS/MS Molecules doi: 10.3390/molecules24132410 Authors: Cuiting Wu Xin Wang Ming Xu Youping Liu Xin Di A novel strategy was developed to identify hepatotoxic compounds in traditional Chinese medicines (TCMs). It is based on the exposure of HL-7702 cells to a TCM extract, followed by the identification and further determination...
Sat Jun 29, 2019 03:00
Molecules, Vol. 24, Pages 2411: NFBTA: A Potent Cytotoxic Agent against Glioblastoma Molecules doi: 10.3390/molecules24132411 Authors: Hasan Turkez Flávio Rogério da Nóbrega Ozlem Ozdemir Carlos da Silva Maia Bezerra Filho Reinaldo Nóbrega de Almeida Eduardo Tejera Yunierkis Perez-Castillo Damião Pergentino de Sousa Piplartine (PPL), also known as piperlongumine, is a biologically active alkaloid extracted from the Piper genus which has been found to have highly...
Sat Jun 29, 2019 03:00
Molecules, Vol. 24, Pages 2408: Identification and Characterization of trans-Isopentenyl Diphosphate Synthases Involved in Herbivory-Induced Volatile Terpene Formation in Populus trichocarpa Molecules doi: 10.3390/molecules24132408 Authors: Nathalie D. Lackus Nora P. Petersen Raimund Nagel Axel Schmidt Sandra Irmisch Jonathan Gershenzon Tobias G. Köllner In response to insect herbivory, poplar releases a blend of volatiles that plays important roles in plant defense....
Sat Jun 29, 2019 03:00
Molecules, Vol. 24, Pages 2406: Selective Extraction of ω-3 Fatty Acids from Nannochloropsis sp. Using Supercritical CO2 Extraction Molecules doi: 10.3390/molecules24132406 Authors: Gian Paolo Leone Roberto Balducchi Sanjeet Mehariya Maria Martino Vincenzo Larocca Giuseppe Di Sanzo Angela Iovine Patrizia Casella Tiziana Marino Despina Karatza Simeone Chianese Dino Musmarra Antonio Molino In this article, microalgae Nannochloropsis sp. was used for...
Sat Jun 29, 2019 03:00
Molecules, Vol. 24, Pages 2407: Design, Synthesis and Biological Evaluation of Novel Osimertinib-Based HDAC and EGFR Dual Inhibitors Molecules doi: 10.3390/molecules24132407 Authors: Hang Dong Hao Yin Chunlong Zhao Jiangying Cao Wenfang Xu Yingjie Zhang Herein a novel series of histone deacetylases (HDACs) and epidermal growth factor receptor (EGFR) dual inhibitors were designed and synthesized based on the structure of the approved EGFR inhibitor osimertinib (AZD9291)....
Sat Jun 29, 2019 03:00
Molecules, Vol. 24, Pages 2409: Laboratory Evaluation of Natural and Synthetic Aromatic Compounds as Potential Attractants for Male Mediterranean fruit Fly, Ceratitis capitata Molecules doi: 10.3390/molecules24132409 Authors: Nurhayat Tabanca Marco Masi Nancy D. Epsky Paola Nocera Alessio Cimmino Paul E. Kendra Jerome Niogret Antonio Evidente Ceratitis capitata, the Mediterranean fruit fly, is one of the most serious agricultural pests worldwide responsible for significant...
Sat Jun 29, 2019 03:00
Molecules, Vol. 24, Pages 2405: Synthesis of 6,12-Disubstituted Methanodibenzo[b,f][1,5]dioxocins: Pyrrolidine Catalyzed Self-Condensation of 2′-Hydroxyacetophenones Molecules doi: 10.3390/molecules24132405 Authors: Benedicta Assoah Vesa Riihonen João R. Vale Arto Valkonen Nuno R. Candeias The preparation of unprecedented 6,12-disubstituted methanodibenzo[b,f][1,5]dioxocins from pyrrolidine catalyzed self-condensation of 2′-hydroxyacetophenones is herein described. This method...
Sat Jun 29, 2019 03:00
Molecules, Vol. 24, Pages 2401: Metal Concentration in Muscle and Digestive Gland of Common Octopus (Octopus vulgaris) from Two Coastal Site in Southern Tyrrhenian Sea (Italy) Molecules doi: 10.3390/molecules24132401 Authors: Andrea Ariano Raffaele Marrone Rebecca Andreini Giorgio Smaldone Salvatore Velotto Serena Montagnaro Aniello Anastasio Lorella Severino Octopus vulgaris constitute an important part of most suitable marine resources for human consumption, however,...
Sat Jun 29, 2019 03:00
Molecules, Vol. 24, Pages 2403: Targeting Bacterial Biofilms by the Green Tea Polyphenol EGCG Molecules doi: 10.3390/molecules24132403 Authors: Regine Hengge Bacterial biofilms are multicellular aggregates in which cells are embedded in an extracellular matrix of self-produced biopolymers. Being refractory to antibiotic treatment and host immune systems, biofilms are involved in most chronic infections, and anti-biofilm agents are being searched for urgently. Epigallocatechin-3-gallate...
Sat Jun 29, 2019 03:00
Molecules, Vol. 24, Pages 2402: Synthesis of Fucosyl-Oligosaccharides Using α-l-Fucosidase from Lactobacillus rhamnosus GG Molecules doi: 10.3390/molecules24132402 Authors: Yolanda Escamilla-Lozano Francisco Guzmán-Rodríguez Sergio Alatorre-Santamaría Mariano García-Garibay Lorena Gómez-Ruiz Gabriela Rodríguez-Serrano Alma Cruz-Guerrero Fucosyl-oligosaccharides are natural prebiotics that promote the growth of probiotics in human gut and stimulate the innate immune...
Sat Jun 29, 2019 03:00
Molecules, Vol. 24, Pages 2404: Sphingosine-1-Phosphate Improves the Biological Features of Mouse Bone Marrow-Derived EPCs Partially through PI3K/AKT/eNOS/NO Pathway Molecules doi: 10.3390/molecules24132404 Authors: Xia Wang Enxin Zhan Guohua Lu Qingjie Mu Tianliang Zhang Nana Yang Sphingosine-1-phosphate (S1P), a bioactive sphingolipid, is recognized as a critical regulator in physiological and pathophysiological processes of atherosclerosis (AS). However, the underlying...
Sat Jun 29, 2019 03:00
Molecules, Vol. 24, Pages 2400: Development and Validation of a Method for the Analysis of Bisoprolol and Atenolol in Human Bone Molecules doi: 10.3390/molecules24132400 Authors: Fernandez-Lopez Pellegrini Rotolo Luna Falcon Mancini A method based on gas chromatography–mass spectrometry (GC–MS) is described for the determination of bisoprolol and atenolol in human bone. After the addition of lobivolol as internal standard, pulverized samples were...
Sat Jun 29, 2019 03:00
Molecules, Vol. 24, Pages 2399: An Effective Method of Isolating Honey Proteins Molecules doi: 10.3390/molecules24132399 Authors: Aleksandra Bocian Justyna Buczkowicz Marcin Jaromin Konrad Kamil Hus Jaroslav Legáth Honey is a natural sweetener composed mostly of sugars, but it contains also pollen grains, proteins, free amino acids, and minerals. The amounts and proportions of these components depend on the honey type and bee species. Despite the low content of honey protein,...
Sat Jun 29, 2019 03:00
Molecules, Vol. 24, Pages 2398: Flavonoids from Morus alba L. Leaves: Optimization of Extraction by Response Surface Methodology and Comprehensive Evaluation of Their Antioxidant, Antimicrobial, and Inhibition of α-Amylase Activities through Analytical Hierarchy Process Molecules doi: 10.3390/molecules24132398 Authors: Hao Cui Tenghui Lu Mingxin Wang Xintong Zou Yang Zhang Xiudong Yang Yao Dong Hongli Zhou To explore the flavonoids from Morus alba L. leaves (MLF),...
Fri Jun 28, 2019 03:00
Molecules, Vol. 24, Pages 2396: Long-Term Effect of Ultraviolet Irradiation on Poly(vinyl chloride) Films Containing Naproxen Diorganotin(IV) Complexes Molecules doi: 10.3390/molecules24132396 Authors: Angham G. Hadi Emad Yousif Gamal A. El-Hiti Dina S. Ahmed Khudheyer Jawad Mohammad Hayal Alotaibi Hassan Hashim As poly(vinyl chloride) (PVC) photodegrades with long-term exposure to ultraviolet radiation, it is desirable to develop methods that enhance the photostability...
Fri Jun 28, 2019 03:00
Molecules, Vol. 24, Pages 2395: Mesoporous Silica-Based Materials for Electronics-Oriented Applications Molecules doi: 10.3390/molecules24132395 Authors: Łukasz Laskowski Magdalena Laskowska Neus Vila Mateusz Schabikowski Alain Walcarius Electronics, and nanoelectronics in particular, represent one of the most promising branches of technology. The search for novel and more efficient materials seems to be natural here. Thus far, silicon-based devices have been monopolizing...
Fri Jun 28, 2019 03:00
Molecules, Vol. 24, Pages 2397: Direct Bioelectricity Generation from Sago Hampas by Clostridium beijerinckii SR1 Using Microbial Fuel Cell Molecules doi: 10.3390/molecules24132397 Authors: Mohd Azwan Jenol Mohamad Faizal Ibrahim Ezyana Kamal Bahrin Seung Wook Kim Suraini Abd-Aziz Microbial fuel cells offer a technology for simultaneous biomass degradation and biological electricity generation. Microbial fuel cells have the ability to utilize a wide range of biomass including...
Fri Jun 28, 2019 03:00
Molecules, Vol. 24, Pages 2394: Design, Synthesis, and Biological Application of Novel Photoaffinity Probes of Dihydropyridine Derivatives, BAY R3401 Molecules doi: 10.3390/molecules24132394 Authors: Liying Zhang Zhiwei Yan Youde Wang Chengjun Song Guangxin Miao To explore the molecular mechanisms of BAY R3401, four types of novel photoaffinity probes bearing different secondary tags were synthesized. Their potency for glycogenolysis was evaluated in primary human liver HL-7702...
Fri Jun 28, 2019 03:00
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